SCHEMBL28845393

SCHEMBL28845393

Cc1cnc(N)nc1-c1ccc(Nc2ccnc(N)n2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 11/20 0.56
BCL6 P41182 1/20 0.55
CA12 O43570 1/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA6 P23280 1/20 0.51
CA5A P35218 1/20 0.51
CA7 P43166 1/20 0.51
CA9 Q16790 1/20 0.51
CA14 Q9ULX7 1/20 0.51
CA5B Q9Y2D0 1/20 0.51
KCNH2 Q12809 1/20 0.49
SCN9A Q15858 1/20 0.49
CDC7 O00311 1/20 0.48
MAPKAPK2 P49137 6/20 0.47
CCNE1 P24864 1/20 0.45
CDK2 P24941 1/20 0.45
HTR3E A5X5Y0 1/20 0.45
HTR3B O95264 1/20 0.45
HTR3A P46098 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29808789 1.00 ROCK1 (0.56) ROCK1BCL6CA12CA1CA2
SCHEMBL29809026 0.90 KCNH2 (0.45) ROCK1BCL6CA12CA1CA2
SCHEMBL21121005 0.90 KCNH2 (0.45) ROCK1BCL6CA12CA1CA2
SCHEMBL29809036 0.89 INSR (0.48) ROCK1BCL6CA12CA1CA2
SCHEMBL21163904 0.89 INSR (0.48) ROCK1BCL6CA12CA1CA2
SCHEMBL21163558 0.85 ABL1 (0.45) ROCK1BCL6CA12CA1CA2
SCHEMBL29809040 0.85 ABL1 (0.45) ROCK1BCL6CA12CA1CA2
SCHEMBL21163561 0.84 PAK4 (0.41) ROCK1BCL6
SCHEMBL29808697 0.84 PAK4 (0.41) ROCK1BCL6
SCHEMBL21163559 0.83 HRH4 (0.55) ROCK1BCL6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111065635-B Novel pyrimidine derivatives as MTH1 inhibitors 无锡安万生物科技有限公司 2022-07-22 CN claimed