SCHEMBL29808697

SCHEMBL29808697

Cc1cnc(N)nc1-c1ccc(Nc2ccnc(NC3CC3)n2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAK4 O96013 1/20 0.41
PAK1 Q13153 1/20 0.41
ROCK1 Q13464 4/20 0.40
CDK9 P50750 2/20 0.40
CDK7 P50613 1/20 0.40
SYK P43405 1/20 0.39
MAPK1 P28482 3/20 0.39
CCNT1 O60563 1/20 0.39
FLT3 P36888 1/20 0.39
BCL6 P41182 1/20 0.39
MEN1 O00255 2/20 0.38
NPC1 O15118 2/20 0.38
LMNA P02545 2/20 0.38
MAPT P10636 2/20 0.38
RAB9A P51151 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 1/20 0.38
AURKA O14965 1/20 0.38
ALOX12 P18054 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21163561 1.00 PAK4 (0.41) PAK4PAK1ROCK1CDK9CDK7
SCHEMBL21164015 0.96 AURKB (0.42) PAK4PAK1ROCK1MAPK1BCL6
SCHEMBL21163904 0.85 INSR (0.48) ROCK1SYKMAPK1BCL6MEN1
SCHEMBL29809036 0.85 INSR (0.48) ROCK1SYKMAPK1BCL6MEN1
SCHEMBL28845393 0.84 ROCK1 (0.56) ROCK1BCL6
SCHEMBL29808789 0.84 ROCK1 (0.56) ROCK1BCL6
SCHEMBL21163558 0.82 ABL1 (0.45) ROCK1CDK7SYKMAPK1FLT3
SCHEMBL29809040 0.82 ABL1 (0.45) ROCK1CDK7SYKMAPK1FLT3
SCHEMBL29808929 0.81 PLK1 (0.40) ROCK1SYKMAPK1FLT3MEN1
SCHEMBL21163559 0.80 HRH4 (0.55) ROCK1SYKMAPK1BCL6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111065635-B Novel pyrimidine derivatives as MTH1 inhibitors 无锡安万生物科技有限公司 2022-07-22 CN disclosed