SCHEMBL28845641

SCHEMBL28845641

O=C(Nc1cccc([N+](=O)[O-])c1)c1cccc(Nc2ccnc3cc(C(F)(F)F)ccc23)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 2/20 0.55
DNMT1 P26358 2/20 0.54
DNMT3A Q9Y6K1 2/20 0.54
MAPT P10636 4/20 0.53
KMT2A Q03164 4/20 0.53
MEN1 O00255 3/20 0.53
POLB P06746 1/20 0.53
BLM P54132 1/20 0.53
LMNA P02545 2/20 0.50
USP2 O75604 1/20 0.50
NPC1 O15118 1/20 0.50
ALDH1A1 P00352 1/20 0.50
NFKB1 P19838 1/20 0.50
RAB9A P51151 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
BRAF P15056 1/20 0.49
AKR1B1 P15121 1/20 0.48
AKR1C4 P17516 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29809959 1.00 RXFP1 (0.55) RXFP1DNMT1DNMT3AMAPTKMT2A
SCHEMBL28845675 0.87 DNMT1 (0.68) RXFP1DNMT1DNMT3AMAPTLMNA
SCHEMBL28845676 0.87 RXFP1 (0.59) RXFP1DNMT1NPC1RAB9A
SCHEMBL29809944 0.87 RXFP1 (0.59) RXFP1DNMT1NPC1RAB9A
SCHEMBL28845693 0.85 MEN1 (0.61) RXFP1DNMT1DNMT3AMAPTKMT2A
SCHEMBL29809955 0.85 MEN1 (0.61) RXFP1DNMT1DNMT3AMAPTKMT2A
SCHEMBL28845688 0.83 DNMT1 (0.63) RXFP1DNMT1DNMT3ALMNAAURKA
SCHEMBL29200469 0.82 GAK (0.55) DNMT1DNMT3ANPC1AKR1C3AKR1C2
SCHEMBL13335917 0.81 DNMT1 (0.69) DNMT1DNMT3AMAPTKMT2AMEN1
SCHEMBL28845668 0.81 GAA (0.60) DNMT1DNMT3AMAPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114773267-B [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2024-01-26 CN claimed
CN-114773267-A [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2022-07-22 CN claimed
CN-114773267-B [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2024-01-26 CN disclosed
CN-114773267-A [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2022-07-22 CN disclosed