SCHEMBL29200469

SCHEMBL29200469

CC(=O)c1cccc(Nc2ccnc3cc(C(F)(F)F)ccc23)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAK O14976 2/20 0.55
GSK3A P49840 4/20 0.54
GSK3B P49841 4/20 0.54
AKR1C3 P42330 1/20 0.52
AKR1C2 P52895 1/20 0.52
NPC1 O15118 1/20 0.52
CLK4 Q9HAZ1 4/20 0.52
KDR P35968 3/20 0.52
PRKD3 O94806 2/20 0.52
MAP4K4 O95819 2/20 0.52
AURKB Q96GD4 2/20 0.52
PRKD2 Q9BZL6 2/20 0.52
HIPK4 Q8NE63 2/20 0.52
SRPK1 Q96SB4 2/20 0.52
MAP3K20 Q9NYL2 2/20 0.52
MARK3 P27448 1/20 0.52
MAPKAPK2 P49137 1/20 0.52
PRKCZ Q05513 1/20 0.52
PRKAA1 Q13131 1/20 0.52
PAK1 Q13153 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28845693 0.87 MEN1 (0.61) GAKGSK3AGSK3BCLK4KDR
SCHEMBL29809955 0.87 MEN1 (0.61) GAKGSK3AGSK3BCLK4KDR
SCHEMBL28845637 0.86 DNMT1 (0.52) GAKGSK3AGSK3BCLK4KDR
SCHEMBL28845648 0.86 NPSR1 (0.56) GAKGSK3AGSK3BCLK4KDR
SCHEMBL28845675 0.86 DNMT1 (0.68) GAKGSK3AGSK3BNPC1CLK4
SCHEMBL28845679 0.86 GAK (0.50) GAKGSK3AGSK3BAKR1C3AKR1C2
SCHEMBL28845687 0.85 ALDH1A1 (0.57) GAKGSK3AGSK3BCLK4KDR
SCHEMBL28845668 0.84 GAA (0.60) GAKGSK3AGSK3BCLK4KDR
SCHEMBL28845651 0.83 GPR52 (0.54) GAKGSK3AGSK3BCLK4KDR
SCHEMBL4751350 0.83 CYP2D6 (0.58) GAKNPC1DNMT1DNMT3APTK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114773267-B [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2024-01-26 CN claimed