SCHEMBL28845871

SCHEMBL28845871

COC(=O)c1cc(F)c(-c2ccc(N3CCN(C)CC3)cc2)cc1[N+](=O)[O-]

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 8/20 0.67
ALDH1A1 P00352 3/20 0.50
WDR5 P61964 4/20 0.49
PLK1 P53350 1/20 0.46
MAPT P10636 4/20 0.46
LMNA P02545 1/20 0.46
POLB P06746 1/20 0.46
MAPK1 P28482 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.43
HTR6 P50406 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28845823 0.88 SIRT6 (0.69) SIRT6ALDH1A1WDR5PLK1MAPT
SCHEMBL28845819 0.88 SIRT6 (0.50) SIRT6ALDH1A1MAPTLMNAMAPK1
SCHEMBL29891093 0.81 WDR5 (0.59) SIRT6ALDH1A1WDR5MAPTLMNA
SCHEMBL28900077 0.81 SIRT6 (0.81) SIRT6ALDH1A1PLK1MAPTMAPK1
SCHEMBL22652232 0.81 SIRT6 (1.00) SIRT6ALDH1A1MAPTMAPK1L3MBTL1
SCHEMBL31739551 0.79 SIRT6 (0.63) SIRT6ALDH1A1WDR5MAPTLMNA
SCHEMBL28845809 0.76 SIRT6 (0.51) SIRT6ALDH1A1MAPTLMNAMAPK1
SCHEMBL1890774 0.73 SIRT6 (0.61) SIRT6ALDH1A1WDR5MAPTLMNA
SCHEMBL5054829 0.73 MAPT (0.64) SIRT6ALDH1A1MAPTMAPK1L3MBTL1
SCHEMBL5624466 0.73 SIRT6 (0.76) SIRT6ALDH1A1MAPTLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109734674-B Aniline WDR5 protein-protein interaction inhibitor and preparation method and application thereof 中国药科大学 2022-08-26 CN disclosed