SCHEMBL288460

SCHEMBL288460

Cc1nc(-c2ccc(-c3ccc4ccccc4c3)s2)sc1C(=O)NCCN1CCOCC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C19 P33261 1/20 0.55
CD274 Q9NZQ7 2/20 0.52
ALDH1A1 P00352 4/20 0.50
HSD17B10 Q99714 2/20 0.50
CYP3A4 P08684 1/20 0.50
MAPT P10636 1/20 0.50
CYP2C9 P11712 1/20 0.50
ACHE P22303 1/20 0.50
HPGDS O60760 1/20 0.50
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
TSHR P16473 1/20 0.49
LMNA P02545 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
PRF1 P14222 2/20 0.48
HPGD P15428 3/20 0.47
KDM4E B2RXH2 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290307 0.86 CD274 (0.61) CYP1A2CYP2D6CYP2C19CD274ALDH1A1
SCHEMBL298546 0.82 MAPK1 (0.56) CYP1A2ALDH1A1HSD17B10CYP3A4MAPT
SCHEMBL21763579 0.79 ERN1 (0.51) CYP1A2CYP2D6CYP2C19CD274ALDH1A1
SCHEMBL3403357 0.77 DRD3 (0.49) CYP1A2CYP2D6CYP3A4TSHRLMNA
SCHEMBL12675177 0.76 ERN1 (0.65) CYP1A2CD274ALDH1A1HSD17B10CYP3A4
SCHEMBL23956927 0.76 CD274 (0.52) CYP1A2CYP2D6CYP2C19CD274ALDH1A1
SCHEMBL23956924 0.75 TSHR (0.49) CYP1A2CYP2C19CD274ALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL29217421 0.75 TSHR (0.48) CYP1A2CYP2C19CD274ALDH1A1HSD17B10
SCHEMBL289866 0.74 SMN1; SMN2 (0.59) ALDH1A1MAPTLMNASMN1; SMN2HPGD
SCHEMBL3398394 0.74 KDM4E (0.54) CYP1A2CYP2D6ALDH1A1HSD17B10CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed