SCHEMBL290307

SCHEMBL290307

Cc1nc(-c2ccc(-c3cc4ccccc4s3)s2)sc1C(=O)NCCN1CCOCC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 1/20 0.61
LMNA P02545 3/20 0.53
CYP1A2 P05177 2/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C19 P33261 1/20 0.48
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
HPGDS O60760 1/20 0.46
HSD17B10 Q99714 3/20 0.46
PARP1 P09874 1/20 0.45
KMT2A Q03164 2/20 0.45
TSHR P16473 1/20 0.45
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
POLB P06746 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
IKBKB O14920 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL288460 0.86 CYP1A2 (0.55) CD274LMNACYP1A2CYP2D6CYP2C19
SCHEMBL298546 0.82 MAPK1 (0.56) LMNACYP1A2KDM4EALDH1A1HPGD
SCHEMBL289905 0.81 HPGD (0.60) CYP1A2CYP2D6CYP2C19KDM4EALDH1A1
SCHEMBL23956927 0.74 CD274 (0.52) CD274LMNACYP1A2CYP2D6CYP2C19
SCHEMBL290238 0.74 SMN1; SMN2 (0.56) KDM4EALDH1A1HPGDSMN1; SMN2KMT2A
SCHEMBL289671 0.74 HTR2C (0.57) LMNAKDM4EALDH1A1SMN1; SMN2KMT2A
SCHEMBL21763579 0.73 ERN1 (0.51) CD274LMNACYP1A2CYP2D6CYP2C19
SCHEMBL14925215 0.73 LMNA (0.56) CD274LMNACYP1A2ALDH1A1HSD17B10
SCHEMBL2787018 0.72 SMN1; SMN2 (0.41) KDM4EALDH1A1HPGDSMN1; SMN2KMT2A
SCHEMBL23956924 0.72 TSHR (0.49) CD274LMNACYP1A2CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed