SCHEMBL21763579

SCHEMBL21763579

Cc1nc(-c2ccc3c(C=O)cccc3c2)sc1C(=O)NCCN1CCOCC1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.51
HPGDS O60760 2/20 0.50
CD274 Q9NZQ7 2/20 0.48
TSHR P16473 1/20 0.47
LMNA P02545 2/20 0.47
ALDH1A1 P00352 4/20 0.46
HSD17B10 Q99714 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 1/20 0.46
MAPT P10636 1/20 0.46
KDM4E B2RXH2 2/20 0.45
HPGD P15428 2/20 0.45
RXFP1 Q9HBX9 1/20 0.44
POLB P06746 1/20 0.44
CYP2C19 P33261 2/20 0.44
PARP1 P09874 1/20 0.44
CYP2D6 P10635 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12675177 0.86 ERN1 (0.65) ERN1HPGDSCD274TSHRLMNA
SCHEMBL23956927 0.79 CD274 (0.52) CD274TSHRLMNAALDH1A1HSD17B10
SCHEMBL288460 0.79 CYP1A2 (0.55) HPGDSCD274TSHRLMNAALDH1A1
SCHEMBL23956924 0.77 TSHR (0.49) HPGDSCD274TSHRLMNAALDH1A1
Hydrochloric Acid SCHEMBL29217421 0.76 TSHR (0.48) HPGDSCD274TSHRLMNAALDH1A1
SCHEMBL3396816 0.75 HPGD (0.57) CD274TSHRLMNAALDH1A1HSD17B10
SCHEMBL290307 0.73 CD274 (0.61) HPGDSCD274TSHRLMNAALDH1A1
SCHEMBL3404510 0.73 HPGD (0.49) CD274LMNAALDH1A1MAPTHPGD
SCHEMBL298546 0.73 MAPK1 (0.56) TSHRLMNAALDH1A1HSD17B10CYP2C9
SCHEMBL3398394 0.72 KDM4E (0.54) LMNAALDH1A1HSD17B10CYP2C9CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496230-B1 IRE-1 ALPHA INHIBITORS FOSUN ORINOVE PHARMATECH INC (CN) 2020-02-26 EP disclosed