SCHEMBL28847217

SCHEMBL28847217

O=C(Nc1ccccc1NC(OCCCCCCCl)c1ccccc1)c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC3 O15379 1/20 0.46
HDAC2 Q92769 1/20 0.46
TP53 P04637 1/20 0.44
EPHX2 P34913 2/20 0.44
ALDH1A1 P00352 3/20 0.44
HTT P42858 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
ALOX15 P16050 1/20 0.44
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
LMNA P02545 1/20 0.43
RAB9A P51151 1/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28847154 0.72 MAPK1 (0.53) MAPTHDAC1HDAC3HDAC2LMNA
SCHEMBL28847140 0.67 MAPT (0.64) MAPTHDAC1HDAC3HDAC2TP53
SCHEMBL10884343 0.67 LMNA (0.74) MAPTALDH1A1L3MBTL1CYP2C9CYP2C19
SCHEMBL31171396 0.67 HDAC3 (0.68) MAPTHDAC1HDAC3HDAC2ALDH1A1
SCHEMBL27726301 0.66 HDAC1 (0.63) MAPTHDAC1HDAC3HDAC2TP53
SCHEMBL11194354 0.66 MAPT (0.74) MAPTTP53ALDH1A1HTTL3MBTL1
SCHEMBL29155474 0.66 LMNA (0.72) MAPTALDH1A1L3MBTL1CYP2C9CYP2C19
SCHEMBL8819152 0.66 KDM4D (0.68) MAPTHDAC1HDAC3HDAC2TP53
SCHEMBL1520536 0.65 HDAC1 (0.70) MAPTHDAC1HDAC3HDAC2TP53
SCHEMBL7251498 0.65 EPHX2 (0.61) HDAC1EPHX2ALDH1A1HTTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109836378-B Sphingomyelin synthase inhibitor, preparation method and application thereof 上海华汇拓医药科技有限公司 2022-09-30 CN claimed
CN-109836378-B Sphingomyelin synthase inhibitor, preparation method and application thereof 上海华汇拓医药科技有限公司 2022-09-30 CN disclosed