SCHEMBL28848043

SCHEMBL28848043

CC(C)c1nn(Br)c2ccccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
ATM Q13315 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PDE5A O76074 6/20 0.37
PDE4B Q07343 6/20 0.37
PDE3A Q14432 4/20 0.37
MIF P14174 2/20 0.37
KMT2A Q03164 2/20 0.37
ADORA1 P30542 2/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
PDE4A P27815 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2738313 0.78 KDM4E (0.49) TSHRMAPK1PDE5APDE4BPDE3A
SCHEMBL13708517 0.77 MPO (0.42) TSHRMAPTMAPK1CASP1CASP7
SCHEMBL14158377 0.77 PDE5A (0.41) TSHRMAPTMAPK1CASP1CASP7
SCHEMBL27371927 0.75 MIF (0.37) TSHRPDE5APDE4BPDE3AMIF
SCHEMBL14158375 0.75 ELANE (0.36) TSHRMAPTPDE5APDE4BPDE3A
SCHEMBL14239447 0.75 ELANE (0.36) TSHRMAPTPDE5APDE4BPDE3A
SCHEMBL14158374 0.75 ELANE (0.36) TSHRMAPTPDE5APDE4BPDE3A
SCHEMBL18993228 0.74 SLC9A1 (0.41) TSHRMAPTCASP1CASP7PDE5A
SCHEMBL15488683 0.74 MPO (0.37) TSHRMAPTMAPK1CASP1CASP7
SCHEMBL18556459 0.74 PDE4B (0.36) TSHRMAPTMAPK1CASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107337659-A Compounds as protein kinase modulators 理森制药股份公司 2017-11-10 CN disclosed
CN-103702989-B Novel compounds as modulators of protein kinases 理森制药股份公司 2017-07-07 CN disclosed