SCHEMBL28848356

SCHEMBL28848356

COc1c([N+](=O)[O-])ccc(N2CCN(C)CC2)c1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 5/20 0.53
MAPT P10636 5/20 0.50
ALDH1A1 P00352 4/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
CYP1A2 P05177 2/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
LMNA P02545 2/20 0.49
POLB P06746 1/20 0.47
MAPK1 P28482 2/20 0.47
TP53 P04637 1/20 0.47
TSHR P16473 1/20 0.47
HIF1A Q16665 1/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
USP2 O75604 1/20 0.47
S100A4 P26447 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2209087 0.86 ALDH1A1 (0.47) SIRT6MAPTALDH1A1SMN1; SMN2LMNA
SCHEMBL521342 0.85 MAPT (0.50) MAPTALDH1A1SMN1; SMN2LMNAPOLB
SCHEMBL3315189 0.85 MAPT (0.54) MAPTALDH1A1LMNAMAPK1MEN1
SCHEMBL16513957 0.84 MAPT (0.56) SIRT6MAPTALDH1A1SMN1; SMN2CYP1A2
SCHEMBL29847859 0.84 MAPT (0.56) SIRT6MAPTALDH1A1SMN1; SMN2CYP1A2
SCHEMBL3346768 0.83 ALDH1A1 (0.44) SIRT6MAPTALDH1A1LMNAMAPK1
SCHEMBL30464721 0.82 MAPT (0.54) SIRT6MAPTALDH1A1SMN1; SMN2CYP1A2
SCHEMBL22471527 0.82 MAPT (0.54) SIRT6MAPTALDH1A1SMN1; SMN2CYP1A2
SCHEMBL20367087 0.81 MAPT (0.45) MAPTALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL521625 0.81 MAPT (0.46) MAPTALDH1A1LMNAKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106916112-B Pyrimidine derivative, preparation method and medical application thereof 四川海思科制药有限公司 2019-12-20 CN disclosed
CN-106916112-A Pyrimidine derivatives and preparation method thereof and in application pharmaceutically 四川海思科制药有限公司 2017-07-04 CN disclosed