SCHEMBL28849104

SCHEMBL28849104

COS(=O)(=O)CC1CCN(c2ccccc2)C1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 6/20 0.43
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
DDB1 Q16531 2/20 0.40
CRBN Q96SW2 2/20 0.40
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
ACHE P22303 1/20 0.37
LIPE Q05469 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3841236 0.81 ROCK2 (0.46) ROCK2CA12CA1CA2CA9
SCHEMBL28806018 0.74 ROCK2 (0.46) ROCK2CA12CA1CA2CA9
SCHEMBL28849120 0.74 ROCK2 (0.46) ROCK2CA12CA1CA2CA9
SCHEMBL27470019 0.74 ROCK2 (0.46) ROCK2CA12CA1CA2CA9
SCHEMBL28849106 0.73 DDB1 (0.49) ROCK2CA12CA1CA2CA9
SCHEMBL28849019 0.72 PDE4A (0.46) CA12CA1CA2CA9DDB1
SCHEMBL7576221 0.72 ROCK2 (0.44) ROCK2CA12CA1CA2CA9
SCHEMBL8427476 0.72 HTT (0.47) ROCK2CA12CA1CA2CA9
SCHEMBL15552907 0.71 DDB1 (0.56) ROCK2CA12CA1CA2CA9
SCHEMBL5872162 0.71 MEN1 (0.42) ROCK2ALDH1A1MAPTHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108069952-B Quinolinone compound and application thereof in medicines 广东东阳光药业有限公司 2022-09-27 CN disclosed