SCHEMBL28849019

SCHEMBL28849019

COS(=O)(=O)CC1CC(=O)N(c2ccccc2)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
NPC1 O15118 2/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA13 Q8N1Q1 1/20 0.41
CA14 Q9ULX7 1/20 0.41
CA5B Q9Y2D0 1/20 0.41
ALDH1A1 P00352 3/20 0.41
POLB P06746 2/20 0.41
HPGD P15428 2/20 0.41
USP2 O75604 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9433304 0.84 POLB (0.49) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL7456282 0.80 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL31716545 0.75 BRD4 (0.58) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL2152756 0.74 BPTF (0.61) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL4105055 0.74 POLB (0.51) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL28849021 0.73 NPC1 (0.45) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL12974281 0.72 ALDH1A1 (0.53) ALDH1A1MAPTSMN1; SMN2TP53HTT
SCHEMBL5105230 0.72 GRM2 (0.56) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL28849104 0.72 ROCK2 (0.43) NPC1CA12CA1CA2CA9
SCHEMBL892079 0.70 ALDH1A1 (0.67) NPC1CA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108069952-B Quinolinone compound and application thereof in medicines 广东东阳光药业有限公司 2022-09-27 CN disclosed