SCHEMBL28850690

SCHEMBL28850690

COc1c(C(N)=O)ccc2c1nc(O)n2O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 2/20 0.41
NNMT P40261 1/20 0.41
PARP1 P09874 8/20 0.36
PKN1 Q16512 1/20 0.36
PKN2 Q16513 1/20 0.36
SIK1 P57059 1/20 0.34
SIK2 Q9H0K1 1/20 0.34
SIK3 Q9Y2K2 1/20 0.34
KDM4E B2RXH2 3/20 0.33
HSP90AB1 P08238 1/20 0.33
IKBKB O14920 1/20 0.33
MAPT P10636 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
PLA2G2A P14555 1/20 0.32
ALOX15 P16050 1/20 0.32
PTGS2 P35354 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8524627 0.72 NNMT (0.39) IDH1NNMTPARP1PKN1PKN2
SCHEMBL19437531 0.72 TLR8 (0.45) IDH1NNMTPARP1PKN1PKN2
SCHEMBL11039311 0.72 NNMT (0.52) NNMTPARP1KDM4EIKBKBMAPT
SCHEMBL23529352 0.68 PKN1 (0.45) PARP1PKN1PKN2
SCHEMBL14046288 0.68 PARP1 (0.59) NNMTPARP1KDM4EMAPTTDP1
SCHEMBL27556628 0.68 NNMT (0.44) NNMTPARP1KDM4EIKBKBMAPT
SCHEMBL23552643 0.67 PTGER4 (0.46) PARP1PKN1PKN2
SCHEMBL23552540 0.67 PKN1 (0.47) IDH1PARP1PKN1PKN2
SCHEMBL25095012 0.67 PKN1 (0.47) PARP1PKN1PKN2
SCHEMBL23552645 0.67 PTGER4 (0.45) PARP1PKN1PKN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114981265-A Compound (I) CTXT私人有限公司 2022-08-30 CN disclosed