SCHEMBL28856765

SCHEMBL28856765

CCCC(Cc1ccccc1)C1(C#N)CCNCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.36
SLC6A4 P31645 3/20 0.36
SLC6A3 Q01959 1/20 0.36
MAOB P27338 3/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
HIF1A Q16665 1/20 0.35
TACR1 P25103 1/20 0.33
SIGMAR1 Q99720 3/20 0.33
OPRM1 P35372 2/20 0.33
MME P08473 2/20 0.32
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7522574 0.79 SLC6A2 (0.38) SLC6A2SLC6A4SLC6A3MEN1ALDH1A1
SCHEMBL27624000 0.69 SIGMAR1 (0.42) MAOBMEN1TSHRKMT2ASIGMAR1
SCHEMBL4749321 0.68 USP2 (0.44) SLC6A2SLC6A4MEN1CYP2C9TSHR
SCHEMBL6999690 0.66 USP2 (0.39) SLC6A2SLC6A4MEN1ALDH1A1CYP2C9
SCHEMBL736076 0.65 CYP2C9 (0.42) SLC6A2SLC6A4SLC6A3MAOBMEN1
SCHEMBL8569331 0.65 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3SIGMAR1MME
SCHEMBL11152854 0.65 MAOB (0.42) SLC6A2SLC6A4SLC6A3MAOBSIGMAR1
Hydrochloric Acid SCHEMBL4772769 0.64 MEN1 (0.41) SLC6A2SLC6A4SLC6A3MAOBMEN1
Hydrochloric Acid SCHEMBL22719342 0.63 MEN1 (0.41) SLC6A2SLC6A4SLC6A3MAOBMEN1
SCHEMBL14905909 0.63 MEN1 (0.41) SLC6A2SLC6A4SLC6A3MAOBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922388-A Compounds and compositions for inhibiting SHP2 activity 诺华股份有限公司 2018-04-17 CN disclosed
CN-107787323-A For suppressing the compound and composition of SHP2 activity 诺华股份有限公司 2018-03-09 CN disclosed