SCHEMBL4749321

SCHEMBL4749321

N#CC1(C(c2ccccc2)c2ccccc2)CCNCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 4/20 0.44
CYP2D6 P10635 3/20 0.44
CYP2C9 P11712 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C19 P33261 1/20 0.42
OPRM1 P35372 2/20 0.41
OPRD1 P41143 2/20 0.41
TP53 P04637 1/20 0.39
ALOX15 P16050 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TSHR P16473 2/20 0.36
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SIGMAR1 Q99720 1/20 0.35
HTR2A P28223 1/20 0.35
TRPA1 O75762 1/20 0.34
HSD17B10 Q99714 1/20 0.34
OPRL1 P41146 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6999690 0.79 USP2 (0.39) USP2CYP2D6CYP2C9CYP1A2CYP3A4
SCHEMBL7363061 0.75 USP2 (0.50) USP2CYP2D6CYP2C9CYP1A2CYP3A4
SCHEMBL4749593 0.72 USP2 (0.47) USP2CYP2D6CYP2C9CYP1A2CYP3A4
SCHEMBL1586585 0.69 USP2 (0.39) USP2CYP2D6CYP2C9CYP1A2CYP3A4
SCHEMBL28856765 0.68 SLC6A2 (0.36) CYP2D6CYP2C9CYP2C19OPRM1MEN1
SCHEMBL3360485 0.68 TRPA1 (0.38) CYP2D6OPRM1OPRD1TSHRTRPA1
SCHEMBL2436694 0.68 TRPA1 (0.38) CYP2D6OPRM1OPRD1TSHRTRPA1
SCHEMBL187469 0.68 OPRM1 (0.55) OPRM1OPRD1MEN1KMT2AHTR2A
SCHEMBL4746204 0.68 USP2 (0.44) USP2CYP2D6CYP2C9CYP1A2CYP3A4
SCHEMBL22719169 0.67 SLC6A2 (0.35) SLC6A2SLC6A4SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008124582-A1 RENIN INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-10-16 WO disclosed