SCHEMBL28857481

SCHEMBL28857481

C[C](C)Cn1cc(CC#N)c2cc(Br)ccc21

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KRAS P01116 4/20 0.54
SMN1; SMN2 Q16637 2/20 0.48
GAA P10253 1/20 0.48
CSNK2A1 P68400 2/20 0.43
NPSR1 Q6W5P4 1/20 0.41
IDO1 P14902 3/20 0.38
AKR1A1 P14550 1/20 0.36
AKR1B1 P15121 1/20 0.36
TBXAS1 P24557 1/20 0.36
LMNA P02545 1/20 0.35
CNR2 P34972 2/20 0.35
CNR1 P21554 1/20 0.35
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28206718 0.89 KRAS (0.44) KRASSMN1; SMN2GAACSNK2A1NPSR1
SCHEMBL443715 0.85 KRAS (0.59) KRASSMN1; SMN2GAACSNK2A1NPSR1
SCHEMBL28857440 0.84 CYP2A6 (0.43) KRASSMN1; SMN2GAAAKR1A1AKR1B1
SCHEMBL28247078 0.80 PRMT5 (0.48) SMN1; SMN2TBXAS1
SCHEMBL13035740 0.79 CSNK2A1 (0.48) KRASSMN1; SMN2GAACSNK2A1LMNA
SCHEMBL28857482 0.76 MCL1 (0.42) KRASAKR1A1AKR1B1
SCHEMBL28206298 0.76 ICMT (0.40) KRASAKR1A1AKR1B1CNR2CNR1
SCHEMBL22035559 0.72 KRAS (1.00) KRAS
SCHEMBL26673741 0.70 CSNK2A1 (0.43) KRASSMN1; SMN2CSNK2A1
SCHEMBL26675684 0.70 CSNK2A1 (0.40) KRASSMN1; SMN2GAACSNK2A1AKR1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108341799-A For treating cancer, the novel indole derivative of virus infection and tuberculosis 生物控制术公司 2018-07-31 CN disclosed
CN-104854088-B Novel indole derivatives for the treatment of cancer, viral infections and lung diseases 生物控制术公司 2018-02-16 CN disclosed