SCHEMBL28857482

SCHEMBL28857482

C[C](C)Cn1cc(CC#N)c2ccc(Cl)cc21

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 7/20 0.42
CYP2A6 P11509 1/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.39
AKR1A1 P14550 2/20 0.36
AKR1B1 P15121 2/20 0.36
PTGER1 P34995 2/20 0.35
RAB9A P51151 1/20 0.34
KRAS P01116 1/20 0.34
PRMT5 O14744 1/20 0.33
BCL2L1 Q07817 1/20 0.33
HTR6 P50406 1/20 0.33
USP14 P54578 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28857440 0.89 CYP2A6 (0.43) CYP2A6PTGDR2AKR1A1AKR1B1RAB9A
SCHEMBL28206298 0.84 ICMT (0.40) PTGDR2AKR1A1AKR1B1KRASPRMT5
SCHEMBL28206718 0.84 KRAS (0.44) AKR1A1AKR1B1PTGER1KRASPRMT5
SCHEMBL28178061 0.83 MCL1 (0.45) MCL1PTGDR2AKR1A1AKR1B1PTGER1
SCHEMBL28247078 0.80 PRMT5 (0.48) PTGDR2RAB9APRMT5
SCHEMBL28857481 0.76 KRAS (0.54) AKR1A1AKR1B1KRAS
SCHEMBL15777186 0.70 L3MBTL1 (0.45) MCL1CYP2A6PTGER1HTR6
SCHEMBL29350216 0.70 L3MBTL1 (0.45) MCL1CYP2A6PTGER1HTR6
SCHEMBL6245487 0.70 CYP2A6 (0.48) CYP2A6RAB9AHTR6
SCHEMBL18015855 0.67 KCNH2 (0.46) MCL1PTGER1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108341799-A For treating cancer, the novel indole derivative of virus infection and tuberculosis 生物控制术公司 2018-07-31 CN disclosed
CN-104854088-B Novel indole derivatives for the treatment of cancer, viral infections and lung diseases 生物控制术公司 2018-02-16 CN disclosed