SCHEMBL28859458

SCHEMBL28859458

Cc1cc(CN=O)cc(C(=O)OF)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.41
GRIN2B Q13224 2/20 0.36
MRGPRX4 Q96LA9 2/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
TPMT P51580 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
PARP10 Q53GL7 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32
PRKCA P17252 2/20 0.31
PRKCD Q05655 2/20 0.31
CNR2 P34972 1/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28811339 0.78 TPMT (0.52) SLC7A5NPC1RAB9ATPMTTDP1
SCHEMBL21574901 0.78 PARP10 (0.44) SLC7A5GRIN2BNPC1RAB9ATPMT
SCHEMBL24080830 0.74 PGK1 (0.43) GRIN2BRAB9APGK1PGK2
SCHEMBL28947533 0.70 TSHR (0.46) SLC7A5NPC1RAB9ATPMTTDP1
SCHEMBL28848239 0.70 MAPT (0.36) NPC1RAB9ACA12CA1CA2
SCHEMBL16405265 0.68 SLC7A5 (0.51) SLC7A5TDP1CA12CA1CA2
SCHEMBL27775516 0.67 CA12 (0.39) SLC7A5MRGPRX4TDP1CA12CA1
SCHEMBL16769676 0.67 CA12 (0.58) SLC7A5NPC1CA12CA1CA2
SCHEMBL14143757 0.67 SLC7A5 (0.62) SLC7A5TDP1CA12CA1CA2
SCHEMBL2161045 0.67 SLC7A5 (0.62) SLC7A5TDP1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104379575-B Compounds and compositions for modulating EGFR activity 诺华股份有限公司 2018-04-17 CN disclosed