SCHEMBL28848239

SCHEMBL28848239

Cc1ccc(CN=O)cc1C(=O)OF

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.36
ALOX15 P16050 2/20 0.36
TSHR P16473 2/20 0.36
HPGD P15428 2/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TP53 P04637 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33
NPC1 O15118 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CA12 O43570 2/20 0.31
CA1 P00915 2/20 0.31
CA2 P00918 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28170878 0.80 ALDH1A1 (0.44) ALDH1A1MEN1KMT2ARXRACDC25B
SCHEMBL27999335 0.74 MEN1 (0.49) MAPTALOX15TSHRHPGDTP53
SCHEMBL13268257 0.72 CA12 (0.51) MAPTALOX15TSHRALDH1A1KDM4E
SCHEMBL27966618 0.71 CASP1 (0.44) MAPTALOX15TSHRHPGDALDH1A1
SCHEMBL28859458 0.70 SLC7A5 (0.41) NPC1MEN1KMT2ACA12CA1
SCHEMBL27983812 0.70 ALDH1A1 (0.53) MAPTTSHRHPGDALDH1A1GAA
SCHEMBL28401248 0.69 PKM (0.43) MAPTALOX15TSHRHPGDALDH1A1
SCHEMBL13270403 0.69 SRD5A2 (0.35) NPC1SMN1; SMN2CA12CA1CA2
SCHEMBL27836513 0.69 ALDH1A1 (0.58) MAPTALOX15TSHRHPGDALDH1A1
SCHEMBL28143550 0.69 TSHR (0.36) MAPTALOX15TSHRALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108347943-A HEPATITIS B CORE PROTEIN MODULATORS 组装生物科学股份有限公司 2018-07-31 CN disclosed
CN-108026052-A 5-hydroxyalkyl benzimidazoles as mIDH1 inhibitors 拜耳制药股份公司 2018-05-11 CN disclosed
CN-107949557-A 2 aryl and 2 aralkyl benzimidazoles as mIDH1 inhibitor 拜耳制药股份公司 2018-04-20 CN disclosed
CN-107810176-A N menthyl benzimidazoles compounds as mIDH1 inhibitor 拜耳制药股份公司 2018-03-16 CN disclosed
CN-107108554-A It is used for the phenyl amino benzimidazole of 1 cyclohexyl 2 for treating tumour as MIDH1 inhibitor 拜耳医药股份有限公司 2017-08-29 CN disclosed