SCHEMBL28864474

SCHEMBL28864474

COc1ccccc1-c1ccc(-n2cc(-c3ccccc3)nn2)cc1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
STIM1 Q13586 6/20 0.62
ORAI1 Q96D31 6/20 0.62
PTGS2 P35354 5/20 0.54
PTGS1 P23219 3/20 0.54
OGT O15294 2/20 0.52
CA1 P00915 2/20 0.51
CA2 P00918 2/20 0.51
CA5A P35218 2/20 0.51
CA5B Q9Y2D0 2/20 0.51
CA12 O43570 1/20 0.51
CA9 Q16790 1/20 0.51
ABCG2 Q9UNQ0 1/20 0.50
CYP19A1 P11511 1/20 0.49
MIF P14174 1/20 0.47
AVPR2 P30518 1/20 0.47
OXTR P30559 1/20 0.47
AVPR1A P37288 1/20 0.47
CYP1B1 Q16678 1/20 0.47
DAGLA Q9Y4D2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29946130 0.88 STIM1 (0.56) STIM1ORAI1PTGS2PTGS1OGT
SCHEMBL26628288 0.88 STIM1 (0.56) STIM1ORAI1PTGS2PTGS1OGT
SCHEMBL28864475 0.86 STIM1 (0.54) STIM1ORAI1PTGS2PTGS1OGT
SCHEMBL26628317 0.86 STIM1 (0.85) STIM1ORAI1OGTCA1CA2
SCHEMBL29946211 0.86 STIM1 (0.85) STIM1ORAI1OGTCA1CA2
SCHEMBL26628314 0.82 PTGS2 (0.67) STIM1ORAI1PTGS2PTGS1OGT
SCHEMBL18023900 0.82 PTGS2 (0.58) STIM1ORAI1PTGS2PTGS1OGT
SCHEMBL29946183 0.81 STIM1 (0.85) STIM1ORAI1
SCHEMBL26628283 0.81 STIM1 (0.85) STIM1ORAI1
SCHEMBL2190307 0.81 PTGS2 (0.67) STIM1ORAI1PTGS2PTGS1OGT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115243765-A Biphenyl compounds as SOCE modulators, compositions and uses thereof 皮埃蒙特阿米阿伏伽德罗东方大学 2022-10-25 CN claimed
CN-115243765-A Biphenyl compounds as SOCE modulators, compositions and uses thereof 皮埃蒙特阿米阿伏伽德罗东方大学 2022-10-25 CN disclosed