SCHEMBL2886483

SCHEMBL2886483

CN(C)C1CCN(C(=O)c2cccc(Cn3cnc4ccccc43)c2)C1

nearest known ligand 0.81

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 15/20 0.81
ALDH1A1 P00352 1/20 0.48
CYP11B1 P15538 1/20 0.48
CYP11B2 P19099 1/20 0.48
IDO1 P14902 2/20 0.47
ATR Q13535 1/20 0.47
PDE5A O76074 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2883495 0.89 HRH3 (1.00) HRH3PDE5A
SCHEMBL13085754 0.86 HRH3 (0.76) HRH3ALDH1A1CYP11B1CYP11B2IDO1
SCHEMBL2892498 0.83 HRH3 (0.71) HRH3PDE5A
SCHEMBL1811328 0.82 HRH3 (0.62) HRH3ATR
SCHEMBL2886484 0.82 HRH3 (0.72) HRH3CYP11B1CYP11B2ATR
SCHEMBL2881480 0.81 HRH3 (0.60) HRH3ALDH1A1CYP11B1CYP11B2IDO1
SCHEMBL2887674 0.79 HRH3 (0.78) HRH3ATRPDE5A
SCHEMBL2885714 0.79 HRH3 (0.78) HRH3CYP11B2ATRPDE5A
SCHEMBL2879391 0.79 HRH3 (0.76) HRH3CYP11B2PDE5A
SCHEMBL2884328 0.79 HRH3 (0.76) HRH3CYP11B2PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7820825-B2 N-substituted-azacyclylamines as histamine-3 antagonists WYETH LLC (US) 2010-10-26 US disclosed