SCHEMBL28865712

SCHEMBL28865712

COc1ccc(CN2C(=O)c3ccccc3C2(C)C)cc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.55
CASP3 P42574 2/20 0.53
MDM2 Q00987 4/20 0.52
TP53 P04637 1/20 0.52
PGR P06401 1/20 0.51
MEN1 O00255 1/20 0.49
APAF1 O14727 1/20 0.49
GAA P10253 1/20 0.49
KMT2A Q03164 1/20 0.49
SENP8 Q96LD8 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
SENP6 Q9GZR1 1/20 0.49
KDM4E B2RXH2 1/20 0.49
NR1H3 Q13133 1/20 0.48
CMA1 P23946 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
CHRM5 P08912 1/20 0.46
SCN9A Q15858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2027394 0.85 ALDH1A1 (0.72) ALDH1A1MDM2TP53
SCHEMBL14991625 0.83 MDM2 (0.47) CASP3MDM2TP53CMA1TDP1
SCHEMBL30930026 0.82 RPS6KA2 (0.44) ALDH1A1CASP3MDM2KDM4ECMA1
SCHEMBL18863310 0.82 MDM2 (0.46) ALDH1A1CASP3MDM2CMA1TDP1
SCHEMBL29217149 0.82 RPS6KA2 (0.44) ALDH1A1CASP3MDM2KDM4ECMA1
SCHEMBL1476736 0.82 PARK7 (0.46) CASP3MDM2TP53CMA1TDP1
SCHEMBL14991574 0.82 MDM2 (0.46) ALDH1A1CASP3MDM2CMA1TDP1
SCHEMBL21325286 0.81 MDM2 (0.51) ALDH1A1CASP3MDM2TP53MEN1
SCHEMBL20100132 0.81 MDM2 (0.61) MDM2TP53SCN9A
SCHEMBL21496819 0.79 KDM4E (0.42) ALDH1A1CASP3TP53KDM4ECMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602814-A Pyrrolo-, pyrazolo-, imidazo-pyrimidine and pyridine compounds inhibiting MNK1 and MNK2 效应治疗股份有限公司 2018-09-28 CN disclosed