SCHEMBL28866136

SCHEMBL28866136

CC(C)(Br)Oc1ccccc1C#N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.49
POLB P06746 1/20 0.49
HTR1A P08908 1/20 0.48
ADRA2A P08913 1/20 0.48
ADRA2B P18089 1/20 0.48
MAOA P21397 1/20 0.48
HTR2B P41595 1/20 0.48
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
ALDH1A1 P00352 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
KDM4E B2RXH2 2/20 0.46
TP53 P04637 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TSHR P16473 2/20 0.43
MAPK1 P28482 2/20 0.43
IMPDH2 P12268 1/20 0.43
IMPDH1 P20839 1/20 0.43
HPGD P15428 1/20 0.42
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2154632 0.86 GAA (0.50) GAAPOLBHTR1AADRA2AADRA2B
SCHEMBL103547 0.78 GAA (0.46) GAAPOLBHTR1AADRA2AADRA2B
SCHEMBL11568266 0.78 GAA (0.46) GAAPOLBHTR1AADRA2AADRA2B
SCHEMBL3813926 0.77 HTR1A (0.52) GAAPOLBHTR1AADRA2AADRA2B
SCHEMBL1070157 0.76 POLB (0.45) GAAPOLBHTR1AADRA2AADRA2B
Boric Acid SCHEMBL27921249 0.75 HTR1A (0.42) GAAPOLBHTR1AADRA2AADRA2B
SCHEMBL11244858 0.75 POLB (0.41) GAAPOLBHTR1AADRA2AADRA2B
SCHEMBL973234 0.74 ALDH1A1 (0.54) GAAPOLBHTR1AADRA2AADRA2B
SCHEMBL11748737 0.74 ALDH1A1 (0.54) GAAPOLBHTR1AADRA2AADRA2B
SCHEMBL29182356 0.74 GAA (0.43) GAAPOLBHTR1AADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108863850-A Biaryl base class compound and its preparation method and application 复旦大学 2018-11-23 CN disclosed