SCHEMBL28868007

SCHEMBL28868007

CCn1ccc2c(C(=O)OBr)cccc21

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.50
LMNA P02545 3/20 0.43
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP19A1 P11511 1/20 0.39
CNR2 P34972 7/20 0.39
GAA P10253 1/20 0.39
CNR1 P21554 6/20 0.38
KMT2A Q03164 1/20 0.37
BRD4 O60885 1/20 0.37
SYK P43405 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13824516 0.87 NR4A2 (0.67) NR4A2LMNAALDH1A1SMN1; SMN2GAA
SCHEMBL5761906 0.81 CYP19A1 (0.51) NR4A2LMNAALDH1A1SMN1; SMN2CYP19A1
SCHEMBL28264481 0.81 NR4A2 (0.76) NR4A2LMNAALDH1A1SMN1; SMN2CNR2
SCHEMBL28265649 0.80 TUBB4A (0.52) NR4A2LMNAALDH1A1KMT2A
SCHEMBL28264524 0.77 TDP1 (0.36) NR4A2CYP19A1KMT2ABRD4
SCHEMBL4395116 0.74 HTR2C (0.49) NR4A2LMNA
SCHEMBL28264498 0.74 PDE4B (0.39) NR4A2LMNAALDH1A1SMN1; SMN2KMT2A
SCHEMBL2593643 0.73 NR4A2 (0.53) NR4A2LMNASMN1; SMN2GAACNR1
SCHEMBL15999018 0.72 NR4A2 (0.52) NR4A2LMNAALDH1A1SMN1; SMN2GAA
SCHEMBL1586664 0.72 NR4A2 (0.52) NR4A2LMNASMN1; SMN2CNR2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109153643-A Substituted indole MCL-1 inhibitors 范德比尔特大学 2019-01-04 CN disclosed