SCHEMBL28868525

SCHEMBL28868525

CC(C)(C)OC(=O)N1CC2(CN(Cc3ccnc(Br)c3F)C2)C1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RORC P51449 3/20 0.45
GPR119 Q8TDV5 5/20 0.43
PARP1 P09874 1/20 0.37
AOC3 Q16853 1/20 0.37
CD274 Q9NZQ7 3/20 0.36
PDCD1LG2 Q9BQ51 1/20 0.36
PDCD1 Q15116 2/20 0.35
SCD5 Q86SK9 1/20 0.35
EGLN2 Q96KS0 1/20 0.35
EIF2AK4 Q9P2K8 2/20 0.35
FAAH O00519 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23850069 0.76 RORC (0.48) RORCGPR119CD274PDCD1LG2
SCHEMBL27253377 0.75 RORC (0.56) RORCPARP1
SCHEMBL30620505 0.75 RORC (0.53) RORCPARP1
SCHEMBL23003391 0.75 CYP3A4 (0.52) RORCGPR119
SCHEMBL28868549 0.74 CD274 (0.35) CD274PDCD1LG2PDCD1
SCHEMBL23850532 0.73 RORC (0.55) RORCPARP1
SCHEMBL30013334 0.73 GPR183 (0.54) RORCGPR119
SCHEMBL19173661 0.72 RORC (0.53) RORCGPR119OPRD1OPRK1
SCHEMBL29669150 0.71 RORC (0.48) RORCGPR119CD274PDCD1LG2PDCD1
SCHEMBL20238623 0.71 RORC (0.48) RORCGPR119CD274PDCD1LG2PDCD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232109-A PD-1/PD-L1 small molecule inhibitor and application thereof in medicines 广东东阳光药业有限公司 2022-10-25 CN disclosed