SCHEMBL28868549

SCHEMBL28868549

CC1(O)CN(Cc2ccnc(Br)c2F)C1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 9/20 0.35
PDCD1 Q15116 6/20 0.35
SCN1A P35498 1/20 0.33
SCN5A Q14524 1/20 0.33
SCN8A Q9UQD0 1/20 0.33
LTA4H P09960 2/20 0.32
PDCD1LG2 Q9BQ51 3/20 0.31
TLR7 Q9NYK1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29225552 0.77 ALDH1A1 (0.45)
SCHEMBL28868640 0.77 CD274 (0.44) CD274PDCD1PDCD1LG2
SCHEMBL28957010 0.74 CD274 (0.36) CD274PDCD1PDCD1LG2
SCHEMBL28868525 0.74 RORC (0.45) CD274PDCD1PDCD1LG2
SCHEMBL30740137 0.72 CCR5 (0.43) CD274LTA4HPDCD1LG2
SCHEMBL20296352 0.72 CCR5 (0.43) CD274LTA4HPDCD1LG2
SCHEMBL20296354 0.72 CCR5 (0.43) CD274LTA4HPDCD1LG2
SCHEMBL15260080 0.71 LTA4H (0.42) CD274PDCD1LTA4HTLR7
SCHEMBL27042898 0.71 CYP3A4 (0.41)
SCHEMBL30021389 0.70 CYP2D6 (0.49) LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232109-A PD-1/PD-L1 small molecule inhibitor and application thereof in medicines 广东东阳光药业有限公司 2022-10-25 CN disclosed