SCHEMBL28869825

SCHEMBL28869825

COC(=O)c1ccc(NC(=O)Cc2c[nH]c3ccccc23)cc1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.64
RAB9A P51151 3/20 0.62
GPR84 Q9NQS5 2/20 0.61
ALDH1A1 P00352 3/20 0.60
MAPT P10636 4/20 0.59
NPC1 O15118 1/20 0.59
HDAC1 Q13547 3/20 0.58
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
LMNA P02545 1/20 0.53
STAT3 P40763 1/20 0.53
HSD17B10 Q99714 1/20 0.53
CYP1A2 P05177 1/20 0.53
POLB P06746 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27333421 0.90 HRH3 (0.63) HRH3RAB9AALDH1A1MAPTNPC1
SCHEMBL28869820 0.87 GPR84 (0.61) HRH3RAB9AGPR84ALDH1A1MAPT
SCHEMBL28373785 0.86 MAPT (0.67) HRH3RAB9AALDH1A1MAPTNPC1
SCHEMBL18229439 0.85 HRH3 (0.77) HRH3RAB9AALDH1A1MAPTHDAC1
SCHEMBL17912677 0.85 GPR84 (0.64) HRH3RAB9AGPR84MAPTNPC1
SCHEMBL18229442 0.85 HRH3 (0.69) HRH3RAB9AALDH1A1MAPTNPC1
SCHEMBL7807900 0.84 HRH3 (0.67) HRH3RAB9AALDH1A1MAPTHDAC1
SCHEMBL31218207 0.84 HRH3 (0.67) HRH3RAB9AALDH1A1MAPTHDAC1
SCHEMBL27333111 0.83 HRH3 (0.67) HRH3RAB9AALDH1A1MAPTHDAC1
SCHEMBL25802387 0.82 HRH3 (0.66) HRH3RAB9AALDH1A1MAPTHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478070-A Compound, pharmaceutical composition and application thereof in field of vasodilation or antiviral 山东第一医科大学(山东省医学科学院) 2023-07-25 CN disclosed
CN-115093359-B Compound, pharmaceutical composition and application thereof in field of vasodilation or antiviral 山东第一医科大学(山东省医学科学院) 2023-06-09 CN disclosed
CN-115093359-A Compound, pharmaceutical composition and application of compound and pharmaceutical composition in field of blood vessel expansion or virus resistance 山东第一医科大学(山东省医学科学院) 2022-09-23 CN disclosed