SCHEMBL28869852

SCHEMBL28869852

FC(F)(F)c1ccc(-n2ccc(C(F)(F)F)n2)cn1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.48
RAB9A P51151 4/20 0.48
MAPT P10636 4/20 0.48
NPSR1 Q6W5P4 3/20 0.46
HTT P42858 1/20 0.46
PAX8 Q06710 1/20 0.46
TRPV4 Q9HBA0 1/20 0.46
POLB P06746 1/20 0.43
PRMT6 Q96LA8 1/20 0.41
DHFR P00374 1/20 0.40
KDM4E B2RXH2 1/20 0.39
IDH1 O75874 5/20 0.39
MAPK1 P28482 1/20 0.38
IDH2 P48735 1/20 0.37
CYP3A4 P08684 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30276673 0.85 POLB (0.46) NPC1RAB9AMAPTNPSR1HTT
SCHEMBL31052478 0.85 DHFR (0.44) NPC1RAB9AMAPTNPSR1HTT
SCHEMBL15935031 0.85 HTT (0.46) NPC1RAB9AMAPTNPSR1HTT
SCHEMBL28242208 0.85 TRPV4 (0.42) NPC1RAB9AMAPTNPSR1HTT
SCHEMBL15924259 0.85 TRPV4 (0.42) NPC1RAB9AMAPTNPSR1HTT
SCHEMBL30276683 0.82 MAPT (0.47) NPC1RAB9AMAPTNPSR1HTT
SCHEMBL19311804 0.81 TRPV4 (0.39) NPC1RAB9AMAPTNPSR1HTT
SCHEMBL16043755 0.81 KCNJ1 (0.39) NPC1RAB9AMAPTNPSR1HTT
SCHEMBL287239 0.80 NPC1 (0.53) NPC1RAB9AMAPTNPSR1HTT
SCHEMBL28242163 0.80 DHFR (0.40) TRPV4DHFRIDH1CYP3A4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109476640-A Bicyclic proline compounds 豪夫迈·罗氏有限公司 2019-03-15 CN disclosed
CN-109476628-A Sulfonyl cyclic alkyl amides compound as TRPA1 regulator 豪夫迈·罗氏有限公司 2019-03-15 CN disclosed