SCHEMBL28870331

SCHEMBL28870331

O=c1[nH]ccc2cc(Cl)cc(Br)c12

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 16/20 0.51
CSNK2A1 P68400 1/20 0.41
F7 P08709 1/20 0.40
LTA4H P09960 1/20 0.40
F3 P13726 1/20 0.40
AHR P35869 1/20 0.40
NR4A2 P43354 1/20 0.40
JAK2 O60674 1/20 0.40
RPS6KA3 P51812 1/20 0.40
MELK Q14680 1/20 0.40
STK24 Q9Y6E0 1/20 0.40
PARP1 P09874 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31399012 0.81 CHEK1 (0.54) CHEK1F7LTA4HF3AHR
SCHEMBL25073866 0.80 CHEK1 (0.43) CHEK1AHRJAK2RPS6KA3MELK
SCHEMBL30279145 0.80 CHEK1 (0.43) CHEK1AHRJAK2RPS6KA3MELK
SCHEMBL31227194 0.79 CHEK1 (0.51) CHEK1F7LTA4HF3AHR
SCHEMBL1397681 0.77 CSNK2A1 (0.46) CHEK1CSNK2A1F7LTA4HF3
SCHEMBL25151113 0.75 CHEK1 (0.47) CHEK1CSNK2A1AHRNR4A2JAK2
SCHEMBL31723375 0.73 CHEK1 (0.53) CHEK1CSNK2A1AHRJAK2RPS6KA3
SCHEMBL3117561 0.72 JAK2 (0.61) CHEK1AHRJAK2RPS6KA3MELK
SCHEMBL25317975 0.71 CHEK1 (0.42) CHEK1CSNK2A1JAK2RPS6KA3MELK
SCHEMBL1050400 0.69 CHEK1 (0.49) CHEK1F7LTA4HF3AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111961035-B Compound containing hydroxyisoquinoline structure, pharmaceutical composition and application thereof 南京科技职业学院 2022-11-01 CN disclosed
CN-111961035-A Compound containing hydroxyisoquinoline structure, pharmaceutical composition and application thereof 南京科技职业学院 2020-11-20 CN disclosed