SCHEMBL28870641

SCHEMBL28870641

CC(c1cnccc1C(F)F)C1CC1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 7/20 0.33
ROCK1 Q13464 7/20 0.33
PKN2 Q16513 3/20 0.33
RPS6KA5 O75582 2/20 0.33
LRRK2 Q5S007 2/20 0.33
TP53 P04637 2/20 0.33
CYP3A4 P08684 2/20 0.33
CHUK O15111 1/20 0.33
PRKD3 O94806 1/20 0.33
CDK1 P06493 1/20 0.33
CDK2 P24941 1/20 0.33
LTK P29376 1/20 0.33
CDK8 P49336 1/20 0.33
PRKX P51817 1/20 0.33
CDK5 Q00535 1/20 0.33
PRKCQ Q04759 1/20 0.33
PRKCD Q05655 1/20 0.33
STK3 Q13188 1/20 0.33
PRKG2 Q13237 1/20 0.33
CDC42BPA Q5VT25 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28870639 1.00 ROCK2 (0.33) ROCK2ROCK1PKN2RPS6KA5LRRK2
SCHEMBL28284263 0.79 SLC6A2 (0.31)
SCHEMBL25996380 0.77 RPS6KA3 (0.45) RPS6KA3
SCHEMBL28282710 0.77 MAPT (0.31)
SCHEMBL28284287 0.77 GAA (0.37)
SCHEMBL28282634 0.77 MAPT (0.31)
SCHEMBL28284286 0.77 GAA (0.37)
SCHEMBL28282633 0.77 MAPT (0.31)
SCHEMBL26030475 0.74 RPS6KA3 (0.45) RPS6KA3
SCHEMBL25493980 0.71 TSHR (0.41) TP53HTTTSHRRPS6KA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109415358-A 6-aminopyridin-3-ylthiazoles as ROR gamma t modulators 詹森药业有限公司 2019-03-01 CN disclosed