SCHEMBL28874398

SCHEMBL28874398

FC(F)(F)c1ccc(CSc2nc3ccc(-c4ccccc4)cc3o2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
HPGD P15428 1/20 0.49
CYP2C19 P33261 1/20 0.49
GFER P55789 1/20 0.49
MAPT P10636 4/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
LMNA P02545 2/20 0.46
CASP3 P42574 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
GSK3A P49840 3/20 0.44
GSK3B P49841 3/20 0.44
MAOB P27338 1/20 0.44
L3MBTL1 Q9Y468 3/20 0.43
TSHR P16473 2/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28874437 0.95 CYP1A2 (0.44) CYP1A2CYP2C9HPGDCYP2C19GFER
SCHEMBL28874444 0.92 GSK3B (0.43) CYP1A2CYP2C9HPGDCYP2C19GFER
SCHEMBL28874396 0.91 LMNA (0.47) CYP1A2CYP2C9HPGDCYP2C19GFER
SCHEMBL28874447 0.90 VSIR (0.44) CYP1A2CYP2C9HPGDCYP2C19GFER
SCHEMBL29878676 0.90 VSIR (0.44) CYP1A2CYP2C9HPGDCYP2C19GFER
SCHEMBL28874288 0.89 BCHE (0.41) CYP1A2CYP2C9HPGDCYP2C19GFER
SCHEMBL28874362 0.89 NPC1 (0.46) CYP1A2CYP2C9HPGDCYP2C19GFER
SCHEMBL28874466 0.88 EPHX2 (0.44) CYP1A2CYP2C9HPGDCYP2C19GFER
SCHEMBL28874373 0.88 EPHX2 (0.44) CYP1A2CYP2C9HPGDCYP2C19GFER
SCHEMBL28874291 0.86 GSK3B (0.48) CYP1A2CYP2C9CYP2C19MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115124485-B Sulfoxide-containing benzoxazole derivative, and preparation method and application thereof 中国医学科学院药物研究所 2023-12-15 CN disclosed
CN-115124485-A Benzoxazole derivatives containing sulfoxide as well as preparation method and application thereof 中国医学科学院药物研究所 2022-09-30 CN disclosed