SCHEMBL28874432

SCHEMBL28874432

Clc1ccc2nc(SCc3cccc(-c4ccccc4)c3)oc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.46
NLRP3 Q96P20 1/20 0.46
LMNA P02545 3/20 0.46
KMT2A Q03164 1/20 0.46
CYP1A2 P05177 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
HPGD P15428 1/20 0.45
GFER P55789 1/20 0.45
PTGS1 P23219 2/20 0.45
PTGS2 P35354 2/20 0.45
MAPT P10636 4/20 0.44
TSHR P16473 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ELANE P08246 2/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28874403 0.91 HPGD (0.52) XDHNLRP3LMNAKMT2ACYP1A2
SCHEMBL28874556 0.83 MAPT (0.56) LMNAKMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL28874469 0.82 GSK3B (0.46) HPGDGFERPTGS1PTGS2MAPT
SCHEMBL29878711 0.82 GSK3B (0.50) KMT2APTGS1PTGS2MAPTTSHR
SCHEMBL28874344 0.82 GSK3B (0.50) KMT2APTGS1PTGS2MAPTTSHR
SCHEMBL28874446 0.82 MAPT (0.51) XDHNLRP3LMNAKMT2ACYP1A2
SCHEMBL28874309 0.79 MAPT (0.56) LMNAKMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL28874308 0.78 MAPT (0.52) LMNAKMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL28874335 0.78 MAPT (0.52) LMNAKMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL28874557 0.78 MAPT (0.55) LMNAKMT2ACYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115124485-B Sulfoxide-containing benzoxazole derivative, and preparation method and application thereof 中国医学科学院药物研究所 2023-12-15 CN disclosed
CN-115124485-A Benzoxazole derivatives containing sulfoxide as well as preparation method and application thereof 中国医学科学院药物研究所 2022-09-30 CN disclosed