SCHEMBL28874446

SCHEMBL28874446

COc1cccc(CSc2nc3ccc(Cl)cc3o2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.51
PIK3CB P42338 2/20 0.50
NPSR1 Q6W5P4 3/20 0.49
TSHR P16473 2/20 0.48
MAPK1 P28482 2/20 0.48
CCR2 P41597 1/20 0.48
ALDH1A1 P00352 3/20 0.47
HPGD P15428 2/20 0.47
KMT2A Q03164 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
HSD17B10 Q99714 1/20 0.47
CPB1 P15086 1/20 0.47
LMNA P02545 4/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
TP53 P04637 2/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
MEN1 O00255 1/20 0.46
POLB P06746 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28874432 0.82 XDH (0.46) MAPTNPSR1TSHRHPGDKMT2A
SCHEMBL28874330 0.81 MAPT (0.66) MAPTNPSR1TSHRMAPK1ALDH1A1
SCHEMBL28874556 0.80 MAPT (0.56) MAPTNPSR1TSHRMAPK1ALDH1A1
SCHEMBL29878711 0.79 GSK3B (0.50) MAPTNPSR1TSHRALDH1A1KMT2A
SCHEMBL28874469 0.79 GSK3B (0.46) MAPTNPSR1ALDH1A1HPGDTP53
SCHEMBL28874344 0.79 GSK3B (0.50) MAPTNPSR1TSHRALDH1A1KMT2A
SCHEMBL28874557 0.78 MAPT (0.55) MAPTNPSR1TSHRMAPK1ALDH1A1
SCHEMBL28874316 0.77 XDH (0.43) MAPTPIK3CBMAPK1CCR2LMNA
SCHEMBL29032759 0.77 MAPT (0.64) MAPTNPSR1TSHRMAPK1ALDH1A1
SCHEMBL28874308 0.75 MAPT (0.52) MAPTNPSR1TSHRMAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115124485-B Sulfoxide-containing benzoxazole derivative, and preparation method and application thereof 中国医学科学院药物研究所 2023-12-15 CN disclosed
CN-115124485-A Benzoxazole derivatives containing sulfoxide as well as preparation method and application thereof 中国医学科学院药物研究所 2022-09-30 CN disclosed