SCHEMBL28874469

SCHEMBL28874469

FC(F)(F)c1cccc(CSc2nc3ccc(Cl)cc3o2)c1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.46
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
TP53 P04637 1/20 0.43
P2RY14 Q15391 1/20 0.42
MAPT P10636 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
DAO P14920 1/20 0.42
GFER P55789 2/20 0.41
TOP2A P11388 2/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28874550 0.87 MAPT (0.49) KDM4EALDH1A1HPGDP2RY14MAPT
SCHEMBL28874432 0.82 XDH (0.46) GSK3BKDM4EHPGDMAPTNPSR1
SCHEMBL28874556 0.80 MAPT (0.56) KDM4EALDH1A1HPGDMAPTNPSR1
SCHEMBL29878711 0.79 GSK3B (0.50) GSK3BALDH1A1TP53MAPTNPSR1
SCHEMBL28874444 0.79 GSK3B (0.43) GSK3BALDH1A1GAAHPGDP2RY14
SCHEMBL28874446 0.79 MAPT (0.51) KDM4EALDH1A1HPGDTP53MAPT
SCHEMBL28874344 0.79 GSK3B (0.50) GSK3BALDH1A1TP53MAPTNPSR1
SCHEMBL28874308 0.78 MAPT (0.52) GSK3BKDM4EALDH1A1GAAHPGD
SCHEMBL28874395 0.77 MAPT (0.60) KDM4EALDH1A1HPGDTP53P2RY14
SCHEMBL29878632 0.77 MAPT (0.60) KDM4EALDH1A1HPGDTP53P2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115124485-B Sulfoxide-containing benzoxazole derivative, and preparation method and application thereof 中国医学科学院药物研究所 2023-12-15 CN disclosed
CN-115124485-A Benzoxazole derivatives containing sulfoxide as well as preparation method and application thereof 中国医学科学院药物研究所 2022-09-30 CN disclosed