SCHEMBL28874550

SCHEMBL28874550

FC(F)(F)c1ccc(CSc2nc3ccc(Cl)cc3o2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.49
NPSR1 Q6W5P4 1/20 0.49
DRD2 P14416 1/20 0.46
TOP2A P11388 2/20 0.45
PIK3CG P48736 1/20 0.44
POLB P06746 2/20 0.44
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
GFER P55789 1/20 0.43
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
LMNA P02545 2/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
MBOAT4 Q96T53 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28874395 0.90 MAPT (0.60) MAPTNPSR1DRD2TOP2APOLB
SCHEMBL29878632 0.90 MAPT (0.60) MAPTNPSR1DRD2TOP2APOLB
SCHEMBL28874556 0.88 MAPT (0.56) MAPTNPSR1PIK3CGPOLBCYP2C19
SCHEMBL28874437 0.87 CYP1A2 (0.44) MAPTNPSR1DRD2POLBCYP2C19
SCHEMBL28874469 0.87 GSK3B (0.46) MAPTNPSR1TOP2APOLBHPGD
SCHEMBL28874552 0.86 LMNA (0.47) MAPTNPSR1POLBCYP2C19CYP1A2
SCHEMBL28874308 0.86 MAPT (0.52) MAPTNPSR1PIK3CGPOLBCYP2C19
SCHEMBL28874481 0.85 CYP1A2 (0.43) MAPTNPSR1DRD2POLBCYP2C19
SCHEMBL22524944 0.83 ELANE (0.54) MAPTNPSR1DRD2TOP2ALMNA
SCHEMBL28874557 0.83 MAPT (0.55) MAPTNPSR1PIK3CGPOLBCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115124485-B Sulfoxide-containing benzoxazole derivative, and preparation method and application thereof 中国医学科学院药物研究所 2023-12-15 CN disclosed
CN-114181165-B Heterocyclic sulfoxide compound, preparation method thereof and application thereof in preparation of pseudomonas aeruginosa quorum sensing inhibitor 浙江工业大学 2023-07-11 CN disclosed
CN-115124485-A Benzoxazole derivatives containing sulfoxide as well as preparation method and application thereof 中国医学科学院药物研究所 2022-09-30 CN disclosed
CN-114181165-A Heterocyclic sulfoxide compound, preparation method thereof and application of heterocyclic sulfoxide compound in preparation of pseudomonas aeruginosa quorum sensing inhibitor 浙江工业大学 2022-03-15 CN disclosed