SCHEMBL28875152

SCHEMBL28875152

COc1ccc(CCn2nnc(C(F)(F)F)c2C(=O)O)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.44
GAA P10253 1/20 0.44
PTGER4 P35408 3/20 0.43
AKR1C2 P52895 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
MAPT P10636 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GPR139 Q6DWJ6 1/20 0.41
KDM4E B2RXH2 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B10 Q99714 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
TP53 P04637 1/20 0.40
ALOX15 P16050 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27848902 0.88 AKR1C3 (0.55) AKR1C3PTGER4AKR1C2ALDH1A1MEN1
SCHEMBL20531569 0.86 GAA (0.45) AKR1C3GAAAKR1C2SMN1; SMN2MAPT
SCHEMBL27633657 0.85 MAPT (0.46) AKR1C3GAAPTGER4AKR1C2MAPT
SCHEMBL27830488 0.76 CA1 (0.47) GAASMN1; SMN2MAPTALDH1A1KDM4E
SCHEMBL1412486 0.74 UCHL1 (0.52) AKR1C3GAAPTGER4AKR1C2SMN1; SMN2
SCHEMBL27830557 0.74 PTGER4 (0.53) AKR1C3PTGER4
SCHEMBL20531597 0.73 SMN1; SMN2 (0.49) GAASMN1; SMN2MAPTALDH1A1KDM4E
SCHEMBL22816780 0.72 AKR1C3 (0.48) AKR1C3PTGER4AKR1C2TP53ALOX15
SCHEMBL22815854 0.72 AKR1C3 (0.49) AKR1C3PTGER4AKR1C2MAPTTP53
SCHEMBL939419 0.71 HPGD (0.51) AKR1C3GAAPTGER4AKR1C2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110022875-A Therapeutic inhibiting compound 莱福斯希医药公司 2019-07-16 CN disclosed