SCHEMBL28875992

SCHEMBL28875992

C=CC(=O)Nc1ccc(-c2ccnc(Nc3ccc(N4CCOCC4)cc3)n2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 18/20 1.00
JAK3 P52333 14/20 1.00
JAK1 P23458 8/20 1.00
TYK2 P29597 6/20 1.00
HDAC1 Q13547 2/20 0.69
HDAC6 Q9UBN7 2/20 0.69
HDAC3 O15379 1/20 0.69
NCOR1 O75376 1/20 0.69
HDAC2 Q92769 1/20 0.69
HDAC8 Q9BY41 1/20 0.69
PDGFRB P09619 2/20 0.66
FLT3 P36888 2/20 0.66
IKBKB O14920 1/20 0.66
KIT P10721 1/20 0.66
PDGFRA P16234 1/20 0.66
FLT1 P17948 1/20 0.66
RPS6KB1 P23443 1/20 0.66
FLT4 P35916 1/20 0.66
KDR P35968 1/20 0.66
MAP3K9 P80192 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29813742 1.00 JAK2 (1.00) JAK2JAK3JAK1TYK2HDAC1
SCHEMBL29813541 0.90 JAK2 (1.00) JAK2JAK3JAK1TYK2MAPK8
SCHEMBL28876009 0.90 JAK2 (1.00) JAK2JAK3JAK1TYK2MAPK8
SCHEMBL28875980 0.88 JAK2 (1.00) JAK2JAK3JAK1TYK2HDAC1
SCHEMBL29813618 0.88 JAK2 (1.00) JAK2JAK3JAK1TYK2HDAC1
SCHEMBL4378486 0.88 JAK2 (0.82) JAK2JAK3JAK1TYK2HDAC1
SCHEMBL4390308 0.87 JAK2 (1.00) JAK2JAK3JAK1TYK2HDAC1
SCHEMBL28875997 0.86 JAK2 (0.75) JAK2JAK3JAK1TYK2HDAC1
SCHEMBL4386747 0.85 JAK2 (0.79) JAK2JAK3JAK1TYK2HDAC1
SCHEMBL8082910 0.85 JAK2 (0.81) JAK2JAK3JAK1TYK2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110330484-B Substituted phenyl pyrimidine derivative as JAK kinase inhibitor or pharmaceutically acceptable salt thereof, preparation method and application 中国药科大学 2022-08-26 CN disclosed