SCHEMBL28875997

SCHEMBL28875997

C=CC(=O)Nc1ccc(-c2ccnc(Nc3ccccc3N3CCOCC3)n2)cc1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 17/20 0.75
JAK3 P52333 12/20 0.75
JAK1 P23458 8/20 0.75
TYK2 P29597 6/20 0.75
EGFR P00533 2/20 0.54
HDAC1 Q13547 2/20 0.52
HDAC6 Q9UBN7 2/20 0.52
HDAC3 O15379 1/20 0.52
NCOR1 O75376 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
PDGFRB P09619 2/20 0.50
FLT3 P36888 2/20 0.50
IKBKB O14920 1/20 0.50
KIT P10721 1/20 0.50
PDGFRA P16234 1/20 0.50
FLT1 P17948 1/20 0.50
RPS6KB1 P23443 1/20 0.50
FLT4 P35916 1/20 0.50
KDR P35968 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28876014 0.90 JAK3 (0.77) JAK2JAK3JAK1TYK2EGFR
SCHEMBL28875987 0.89 JAK2 (0.76) JAK2JAK3JAK1TYK2HDAC1
SCHEMBL28875992 0.86 JAK2 (1.00) JAK2JAK3JAK1TYK2EGFR
SCHEMBL29813742 0.86 JAK2 (1.00) JAK2JAK3JAK1TYK2EGFR
SCHEMBL28876026 0.82 JAK3 (0.75) JAK2JAK3JAK1TYK2EGFR
SCHEMBL28556666 0.81 JAK2 (0.77) JAK2JAK3JAK1TYK2PDGFRB
SCHEMBL17287879 0.80 JAK2 (0.56) JAK2JAK3JAK1TYK2HDAC1
SCHEMBL28876006 0.80 JAK2 (0.77) JAK2JAK3JAK1TYK2
Morpholine SCHEMBL28330189 0.79 JAK2 (0.70) JAK2JAK3JAK1TYK2EGFR
SCHEMBL15637731 0.78 JAK2 (0.80) JAK2JAK3JAK1TYK2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110330484-B Substituted phenyl pyrimidine derivative as JAK kinase inhibitor or pharmaceutically acceptable salt thereof, preparation method and application 中国药科大学 2022-08-26 CN disclosed