SCHEMBL28876012

SCHEMBL28876012

C=CC(=O)Nc1cccc(-c2ccnc(Nc3ccc(C4CNCCO4)cc3)n2)c1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 5/20 0.63
JAK2 O60674 4/20 0.63
TYK2 P29597 4/20 0.63
JAK1 P23458 3/20 0.63
EGFR P00533 2/20 0.49
BTK Q06187 1/20 0.49
ITK Q08881 1/20 0.49
PLK1 P53350 1/20 0.49
SLC6A3 Q01959 1/20 0.47
KCNH2 Q12809 1/20 0.47
TAAR1 Q96RJ0 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28875995 0.91 JAK2 (0.61) JAK3JAK2TYK2JAK1SLC6A3
SCHEMBL28876005 0.90 JAK2 (0.64) JAK3JAK2TYK2JAK1PLK1
SCHEMBL28875993 0.84 JAK3 (0.63) JAK3JAK2JAK1EGFRSLC6A3
SCHEMBL28385550 0.84 EGFR (0.61) EGFRSLC6A3KCNH2TAAR1
Morpholine SCHEMBL28328990 0.84 JAK3 (0.73) JAK3JAK2TYK2JAK1EGFR
SCHEMBL28385553 0.82 BTK (0.49) EGFRBTK
SCHEMBL28394043 0.82 EGFR (0.47) EGFRBTKSLC6A3KCNH2TAAR1
SCHEMBL28383433 0.82 EGFR (0.47) EGFRBTKITK
SCHEMBL28385501 0.81 EGFR (0.48) EGFR
SCHEMBL28875983 0.81 JAK2 (0.62) JAK3JAK2TYK2JAK1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110330484-B Substituted phenyl pyrimidine derivative as JAK kinase inhibitor or pharmaceutically acceptable salt thereof, preparation method and application 中国药科大学 2022-08-26 CN disclosed