SCHEMBL28876119

SCHEMBL28876119

Cc1ccccc1-c1ccc2c(c1)C(N1CCN(C)CC1)=Nc1ccccc1N2

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.72
DRD4 P21917 6/20 0.72
CHRM1 P11229 11/20 0.69
DRD3 P35462 4/20 0.69
HRH1 P35367 3/20 0.62
HTR3E A5X5Y0 2/20 0.62
MEN1 O00255 2/20 0.62
HTR3B O95264 2/20 0.62
ABCB11 O95342 2/20 0.62
LMNA P02545 2/20 0.62
ADRB2 P07550 2/20 0.62
CHRM2 P08172 2/20 0.62
CHRM4 P08173 2/20 0.62
HTR1A P08908 2/20 0.62
CHRM5 P08912 2/20 0.62
ADRA2A P08913 2/20 0.62
ADRA2B P18089 2/20 0.62
ADRA2C P18825 2/20 0.62
CHRM3 P20309 2/20 0.62
DRD1 P21728 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28315489 0.86 CHRM1 (0.67) DRD2DRD4CHRM1DRD3HRH1
SCHEMBL14365315 0.85 DRD4 (0.76) DRD2DRD4CHRM1DRD3HRH1
SCHEMBL141020 0.84 DRD2 (1.00) DRD2DRD4CHRM1DRD3HRH1
SCHEMBL29470861 0.84 DRD2 (1.00) DRD2DRD4CHRM1DRD3HRH1
SCHEMBL5557955 0.83 DRD2 (0.74) DRD2DRD4CHRM1DRD3HRH1
Isoclozapine SCHEMBL29822724 0.81 CHRM1 (1.00) DRD2DRD4CHRM1DRD3HRH1
SCHEMBL9094636 0.81 CHRM1 (1.00) DRD2DRD4CHRM1DRD3HRH1
Isoclozapine SCHEMBL140207 0.81 CHRM1 (1.00) DRD2DRD4CHRM1DRD3HRH1
SCHEMBL21234807 0.80 CHRM1 (0.78) DRD2DRD4CHRM1DRD3HRH1
SCHEMBL5918366 0.80 CHRM1 (1.00) DRD2DRD4CHRM1DRD3HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110183387-A Dibenzo diaza * ketone derivatives with anticancer activity and its preparation method and application 新乡医学院 2019-08-30 CN disclosed