SCHEMBL28876830

SCHEMBL28876830

FC(F)(F)c1ccc(C(F)(F)F)c(-n2cccc2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.62
PKM P14618 1/20 0.62
GRIA1 P42261 2/20 0.47
GRIA2 P42262 2/20 0.47
GRIA3 P42263 2/20 0.47
GRIA4 P48058 2/20 0.47
CES2 O00748 2/20 0.43
LMNA P02545 2/20 0.39
MAPK1 P28482 2/20 0.39
MEN1 O00255 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
MAPT P10636 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
PMP22 Q01453 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP2D6 P10635 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
FFAR4 Q5NUL3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29280158 0.79 ALDH1A1 (0.61) ALDH1A1PKMGRIA1GRIA2GRIA3
SCHEMBL25027039 0.79 ALDH1A1 (0.77) ALDH1A1PKMGRIA1GRIA2GRIA3
SCHEMBL31053817 0.79 ALDH1A1 (0.77) ALDH1A1PKMGRIA1GRIA2GRIA3
SCHEMBL2749018 0.79 ALDH1A1 (0.40) ALDH1A1PKMGRIA1GRIA2GRIA3
SCHEMBL12391525 0.77 ALDH1A1 (1.00) ALDH1A1PKMGRIA1GRIA2GRIA3
SCHEMBL13647573 0.77 ALDH1A1 (0.68) ALDH1A1PKMGRIA1GRIA2GRIA3
SCHEMBL30758086 0.77 ALDH1A1 (1.00) ALDH1A1PKMGRIA1GRIA2GRIA3
SCHEMBL16402774 0.74 GRIA1 (0.60) ALDH1A1PKMGRIA1GRIA2GRIA3
SCHEMBL28946277 0.74 ALDH1A1 (0.58) ALDH1A1PKMCES2MAPK1MEN1
SCHEMBL31053823 0.73 ALDH1A1 (0.53) ALDH1A1PKMGRIA1GRIA2GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105408325-B cyanotriazole compounds 大塚制药株式会社 2019-10-22 CN disclosed