SCHEMBL28877856

SCHEMBL28877856

Cn1cc2c(n1)CN(C(=O)O)C2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.42
HDAC2 Q92769 3/20 0.42
NAMPT P43490 2/20 0.38
PDK2 Q15119 1/20 0.33
NOTUM Q6P988 1/20 0.32
KDM1A O60341 1/20 0.32
SLC6A9 P48067 1/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30
TYK2 P29597 1/20 0.30
USP9X Q93008 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26542931 0.86 NOTUM (0.48) HDAC1HDAC2NAMPTPDK2NOTUM
SCHEMBL14861328 0.85 PDK2 (0.45) HDAC1HDAC2NAMPTPDK2NOTUM
SCHEMBL31348202 0.84 HDAC1 (0.44) HDAC1HDAC2NAMPTPDK2NOTUM
SCHEMBL17624333 0.81 HDAC1 (0.42) HDAC1HDAC2NAMPTKDM1ATSHR
SCHEMBL20364273 0.80 PDK2 (0.41) HDAC1HDAC2NAMPTPDK2KDM1A
SCHEMBL26075398 0.80 HDAC1 (0.39) HDAC1HDAC2NAMPTPDK2KDM1A
SCHEMBL15152898 0.78 PDK2 (0.54) PDK2SLC6A9
SCHEMBL15524327 0.77 KDM1A (0.39) KDM1AUSP9X
SCHEMBL25111471 0.75 NOTUM (0.50) NAMPTPDK2NOTUMALDH1A1
SCHEMBL29079151 0.75 PDK2 (0.45) NAMPTPDK2SLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022206730-A1 PYRIMIDOPYRAZINE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-06 WO disclosed
CN-115141202-A Pyrimidopyrazinone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-04 CN disclosed