SCHEMBL28877889

SCHEMBL28877889

CN(C)C(=O)Cn1cc2cc(B3OC(C)(C)C(C)(C)O3)ccc2n1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.39
FFAR1 O14842 1/20 0.35
ROCK1 Q13464 1/20 0.35
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
CCNC P24863 2/20 0.34
CDK8 P49336 2/20 0.34
LIPG Q9Y5X9 7/20 0.33
LPL P06858 6/20 0.33
HIF1A Q16665 1/20 0.32
IRAK4 Q9NWZ3 2/20 0.32
SNCA P37840 1/20 0.32
DGAT1 O75907 1/20 0.32
F2 P00734 1/20 0.32
F11 P03951 1/20 0.32
PRSS1 P07477 1/20 0.32
PRSS2 P07478 1/20 0.32
PRSS3 P35030 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30928610 0.82 IDO1 (0.39) FFAR1ROCK1IDO1TDO2LIPG
SCHEMBL17113584 0.80 LPL (0.41) FFAR1IDO1TDO2LIPGLPL
SCHEMBL23546464 0.80 LPL (0.35) FFAR1IDO1TDO2LIPGLPL
SCHEMBL23638441 0.80 FFAR1 (0.39) FFAR1ROCK1IDO1TDO2LIPG
SCHEMBL31394882 0.78 LPL (0.43) FFAR1IDO1TDO2LIPGLPL
SCHEMBL28877894 0.78 FFAR1 (0.37) FFAR1ROCK1IDO1TDO2LIPG
SCHEMBL17437290 0.78 FFAR1 (0.57) FFAR1IDO1TDO2LIPGLPL
SCHEMBL23633173 0.77 LPL (0.36) FFAR1IDO1TDO2LIPGLPL
SCHEMBL21392369 0.76 CCNC (0.54) FFAR1CCNCCDK8LIPGLPL
SCHEMBL31394025 0.76 IDO1 (0.39) FFAR1ROCK1IDO1TDO2LIPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022206730-A1 PYRIMIDOPYRAZINE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-06 WO disclosed
CN-115141202-A Pyrimidopyrazinone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-04 CN disclosed