SCHEMBL28878014

SCHEMBL28878014

C[Si](C)(C)CCOCn1cc(C(F)(F)F)c2ccc(C(=O)O)cc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.41
PTPN1 P18031 1/20 0.40
NPC1 O15118 1/20 0.39
SLC22A12 Q96S37 3/20 0.38
RORC P51449 2/20 0.37
EGFR P00533 1/20 0.35
IGF1R P08069 1/20 0.35
SRC P12931 1/20 0.35
FLT4 P35916 1/20 0.35
KDR P35968 1/20 0.35
FLT3 P36888 1/20 0.35
EPHB4 P54760 1/20 0.35
TEK Q02763 1/20 0.35
KLKB1 P03952 1/20 0.35
MCL1 Q07820 1/20 0.35
S1PR1 P21453 1/20 0.35
NR1H2 P55055 1/20 0.35
PPARA Q07869 1/20 0.35
NR1H3 Q13133 1/20 0.35
AKR1C3 P42330 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28878087 0.89 NOTUM (0.42) DGAT1PTPN1NPC1EGFRIGF1R
SCHEMBL30166598 0.83 NPC1 (0.41) DGAT1PTPN1NPC1SLC22A12KLKB1
SCHEMBL23855061 0.81 NPC1 (0.40) NPC1SLC22A12EGFRIGF1RSRC
SCHEMBL28878109 0.81 DGAT1 (0.41) DGAT1PTPN1NPC1EGFRIGF1R
SCHEMBL26581238 0.77 NPC1 (0.47) PTPN1NPC1SLC22A12EGFRIGF1R
SCHEMBL23809366 0.75 SLC22A12 (0.45) PTPN1NPC1SLC22A12EGFRIGF1R
SCHEMBL23392592 0.75 MCL1 (0.49) NPC1KLKB1MCL1PPARA
SCHEMBL29653695 0.75 MCL1 (0.49) NPC1KLKB1MCL1PPARA
SCHEMBL25421253 0.74 DGAT1 (0.41) DGAT1PTPN1KLKB1
SCHEMBL23551502 0.72 CNR2 (0.40) NPC1KLKB1MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260180-B Triazole condensed ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2024-05-28 CN disclosed
CN-115260180-A Triazole fused ring containing derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-11-01 CN disclosed