SCHEMBL28878477

SCHEMBL28878477

NNC(=O)c1nc(C(N)=O)cs1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 1/20 0.42
CYP2C19 P33261 1/20 0.42
ACHE P22303 1/20 0.42
ALDH1A1 P00352 4/20 0.38
LMNA P02545 2/20 0.38
PLA2G4A P47712 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
P2RX7 Q99572 4/20 0.36
MAPT P10636 2/20 0.35
HTT P42858 1/20 0.35
GAA P10253 2/20 0.35
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2745784 0.86 HTR2B (0.49) HTR2BCYP2C19ACHEALDH1A1LMNA
SCHEMBL17761019 0.79 CFTR (0.40) HTR2BCYP2C19ACHEPLA2G4A
SCHEMBL12169124 0.79 HTR2B (0.50) HTR2BCYP2C19ACHEALDH1A1LMNA
SCHEMBL17711899 0.78 MAPT (0.50) ALDH1A1LMNAPLA2G4AP2RX7MAPT
SCHEMBL15652132 0.77 HTR2B (0.45) HTR2BCYP2C19ACHEALDH1A1LMNA
SCHEMBL14152154 0.77 HTR2B (0.45) HTR2BCYP2C19ACHEALDH1A1LMNA
SCHEMBL2990831 0.76 NR1I2 (0.52) HTR2BACHEPLA2G4AMAPTGAA
SCHEMBL231752 0.76 GRM5 (0.53) CYP2C19ALDH1A1LMNAP2RX7MAPT
SCHEMBL107709 0.76 S100A4 (0.48) ALDH1A1P2RX7MAPTHTTGAA
SCHEMBL17712058 0.75 PLA2G4A (0.50) HTR2BACHEALDH1A1PLA2G4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108064224-B Amide-substituted thiazoles as modulators of Ror gamma t 詹森药业有限公司 2022-03-29 CN disclosed