SCHEMBL28879474

SCHEMBL28879474

CC(=O)Nc1ccc(-c2ncccc2C(=O)O)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.57
TDP1 Q9NUW8 1/20 0.57
SMN1; SMN2 Q16637 2/20 0.51
HTT P42858 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
TRPV1 Q8NER1 5/20 0.51
KMT2A Q03164 5/20 0.50
PDE10A Q9Y233 1/20 0.50
ALDH1A1 P00352 4/20 0.49
HSD17B10 Q99714 3/20 0.49
HPGD P15428 3/20 0.49
GAA P10253 2/20 0.49
CYP1A2 P05177 2/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
GLA P06280 1/20 0.49
MEN1 O00255 3/20 0.48
POLB P06746 2/20 0.48
PRNP P04156 1/20 0.48
NAPRT Q6XQN6 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002107 0.90 SMN1; SMN2 (0.53) KDM4ESMN1; SMN2HTTL3MBTL1TRPV1
SCHEMBL25359886 0.81 CYP17A1 (0.51) KDM4ETDP1TRPV1
SCHEMBL10726628 0.81 SMN1; SMN2 (0.67) KDM4ETDP1SMN1; SMN2HTTL3MBTL1
SCHEMBL2557875 0.80 KDM4E (0.62) KDM4ETDP1SMN1; SMN2L3MBTL1TRPV1
SCHEMBL14564497 0.80 KDM4E (0.67) KDM4ETDP1SMN1; SMN2L3MBTL1TRPV1
SCHEMBL912675 0.79 KDM4E (0.77) KDM4ETDP1SMN1; SMN2L3MBTL1KMT2A
SCHEMBL31586013 0.79 KDM4E (0.77) KDM4ETDP1SMN1; SMN2L3MBTL1KMT2A
SCHEMBL10094462 0.78 TRPV1 (0.52) KDM4ESMN1; SMN2HTTL3MBTL1TRPV1
SCHEMBL3712467 0.76 KDM4E (0.67) KDM4ETDP1SMN1; SMN2L3MBTL1KMT2A
SCHEMBL31676801 0.76 KDM4E (0.67) KDM4ETDP1SMN1; SMN2L3MBTL1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109608436-B Substituted methyl formyl reagents and methods of using same to improve physicochemical and/or pharmacokinetic properties of compounds 斯法尔制药私人有限公司 2022-10-11 CN disclosed