SCHEMBL9002107

SCHEMBL9002107

CC(=O)Nc1ccc(-c2ncccc2C(=O)c2cccnc2-c2ccc(NC(C)=O)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
HTT P42858 1/20 0.53
TRPV1 Q8NER1 8/20 0.52
KDM4E B2RXH2 3/20 0.50
GAA P10253 2/20 0.50
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
ALDH1A1 P00352 2/20 0.50
HPGD P15428 2/20 0.50
CYP1A2 P05177 1/20 0.50
GLA P06280 1/20 0.50
HSD17B10 Q99714 1/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
PRNP P04156 1/20 0.49
POLB P06746 1/20 0.49
BDKRB1 P46663 1/20 0.48
RORB Q92753 1/20 0.47
NISCH Q9Y2I1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28879474 0.90 KDM4E (0.57) SMN1; SMN2L3MBTL1HTTTRPV1KDM4E
SCHEMBL9002596 0.84 RORB (0.56) SMN1; SMN2L3MBTL1KDM4ENPC1RAB9A
SCHEMBL10726628 0.82 SMN1; SMN2 (0.67) SMN1; SMN2L3MBTL1HTTTRPV1KDM4E
SCHEMBL10094462 0.79 TRPV1 (0.52) SMN1; SMN2L3MBTL1HTTTRPV1KDM4E
SCHEMBL9002488 0.79 RORB (0.48) TRPV1KDM4EGAAALDH1A1HPGD
SCHEMBL9002411 0.79 TRPV1 (0.51) SMN1; SMN2TRPV1KDM4EGAANPC1
SCHEMBL9002089 0.78 NR2E1 (0.46) TRPV1ALDH1A1CYP1A2MEN1KMT2A
SCHEMBL10969548 0.77 RORB (0.60) SMN1; SMN2L3MBTL1KDM4EALDH1A1KMT2A
SCHEMBL8884154 0.76 KDM4E (0.50) SMN1; SMN2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL11350077 0.76 TRPV1 (0.49) SMN1; SMN2L3MBTL1TRPV1KDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5482948-A Pyridyl derivatives and pharmaceutical compositions comprising these compounds DR. KARL THOMAE GMBH (DE) 1996-01-09 US disclosed
US-5286736-A Thromboxane antagonists and thromboxane synthetase inhibitors DR. KARL THOMAE GMBH (DE) 1994-02-15 US disclosed