SCHEMBL28880754

SCHEMBL28880754

Nc1ccccc1NC(=O)c1cc(Br)ccc1Cl

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.66
POLB P06746 1/20 0.66
GAA P10253 1/20 0.66
RECQL P46063 1/20 0.66
RORC P51449 1/20 0.64
TSHR P16473 1/20 0.59
CYP2C19 P33261 3/20 0.57
CYP3A4 P08684 2/20 0.57
CYP2C9 P11712 2/20 0.57
NPSR1 Q6W5P4 1/20 0.57
TP53 P04637 1/20 0.56
KDM4E B2RXH2 3/20 0.55
NPC1 O15118 1/20 0.51
ALDH1A1 P00352 1/20 0.51
RAB9A P51151 1/20 0.51
HDAC1 Q13547 3/20 0.50
HDAC3 O15379 2/20 0.50
HDAC2 Q92769 2/20 0.50
CYP1A2 P05177 1/20 0.50
HPGD P15428 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3509668 0.84 HDAC1 (0.54) MAPTPOLBGAARECQLRORC
SCHEMBL733872 0.83 CYP2C19 (0.58) MAPTPOLBGAARECQLRORC
SCHEMBL28341354 0.83 MAPT (0.70) MAPTPOLBGAARECQLTSHR
SCHEMBL29978583 0.83 MAPT (0.70) MAPTPOLBGAARECQLTSHR
SCHEMBL1283839 0.82 MAPT (0.55) MAPTPOLBGAARECQLRORC
SCHEMBL1624948 0.82 MAPT (0.55) MAPTPOLBGAARECQLRORC
SCHEMBL14671422 0.79 RORC (1.00) MAPTPOLBGAARORCTSHR
SCHEMBL29568686 0.79 RORC (1.00) MAPTPOLBGAARORCTSHR
SCHEMBL28823050 0.78 RORC (0.52) RORCCYP2C19TP53KDM4ENPC1
SCHEMBL641991 0.77 KDM4E (0.69) MAPTGAARORCCYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110494431-B Azacyclo derivative, preparation method and medical application thereof 苏州浦合医药科技有限公司 2022-11-04 CN disclosed
CN-110494431-A Nitrogen heterocycles derivative, preparation method and its medical usage BEIJING YUEZHIKANGTAI BIOMEDICINES CO LTD 2019-11-22 CN disclosed