SCHEMBL28881024

SCHEMBL28881024

CCOC(=O)C1=C(C)NC(C=O)NC1c1cccc(Br)c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.48
DHFR P00374 1/20 0.44
POLB P06746 2/20 0.43
CACNA1B Q00975 1/20 0.42
MAPK1 P28482 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
CACNA1F O60840 2/20 0.40
CACNA1D Q01668 2/20 0.40
CACNA1S Q13698 2/20 0.40
CACNA1C Q13936 2/20 0.40
ABCB1 P08183 1/20 0.40
GAA P10253 2/20 0.40
ALDH1A1 P00352 4/20 0.40
LMNA P02545 1/20 0.39
ALOX12 P18054 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ADORA3 P0DMS8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28345331 0.87 MAPK1 (0.51) KIF11DHFRPOLBCACNA1BMAPK1
SCHEMBL28346142 0.86 HSD17B10 (0.45) DHFRPOLBMAPTGAAALDH1A1
SCHEMBL28346144 0.79 ABCC1 (0.54) MAPK1TP53CACNA1DGAAALDH1A1
SCHEMBL28345988 0.79 MEN1 (0.49) DHFRMAPTGAAALDH1A1LMNA
SCHEMBL5352781 0.78 KIF11 (0.77) KIF11MAPK1GAAALDH1A1SMN1; SMN2
SCHEMBL28342583 0.75 TSHR (0.63) DHFRPOLBMAPK1TP53MAPT
SCHEMBL28349893 0.74 SMN1; SMN2 (0.46) TP53MAPTGAALMNASMN1; SMN2
SCHEMBL3032551 0.73 CACNA1F (0.66) POLBCACNA1BMAPK1MAPTCACNA1F
SCHEMBL27509714 0.73 KMT2A (0.50) DHFRPOLBMAPTCACNA1FCACNA1D
SCHEMBL14413510 0.73 POLB (0.77) POLBMAPTGAAALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108129398-B Synthesis method of 4-halogenated phenyl-5-ethoxycarbonyl-6-methyl-3, 4-dihydropyrimidine-2 (1H) -ketone 大连大学 2020-01-17 CN disclosed